Ucing # | Ngaran produk | Katerangan |
CPD111306 | 7-bromo-2,4,6-trikloro-8-fluoroquinazoline | |
CPD113109 | ARS-1323-Alkuna | ARS-1323-alkuna, saku switch-II (S-IIP) inhibitor |
CPDP801183 | VVD-214;RO7589831;VVD-133214 | VVD-214 mangrupakeun sintétik WRN helikase inhibitor allosteric bisa nepi ka tiwasna. |
CPDP801366 | Inlexisertib;DCC-3116 | DCC-3116 mangrupa inhibitor ULK1/2 oral aktif. |
CPDA601378 | Oranyeu Nonylacridine | |
CPD112537 | 4H-1,3-Dioxolo[4,5-c]pirol-4-asam karboksilat,... | |
CPDP801763 | MC3138 | MC3138 mangrupakeun aktivator SIRT5 selektif. |
CPDP801758 | Chk1-IN-6 | Chk1-IN-6 mangrupakeun potent, selektif, sarta oral bioavailable CHK1 inhibitor calon. |
CPD113410 | NDI-101150 | NDI-101150 mangrupakeun inhibitor potent tur selektif HPK1 (hematopoietic progenitor sél kinase 1). |
CPDA601453 | BMS-986408 | BMS-986408 mangrupakeun oral éféktif dual DGK α / Zeta inhibitor. |
CPDA601445 | AZD0780;EX-A6975;laroprovstatum; laroprovstat | PCSK9-IN-12 mangrupakeun sanyawa heteroaromatic. PCSK9-IN-12 boga pangirut mengikat keur PCSK9 kalawan nilai Kd<200 nM. PCSK9-IN-12 tiasa dianggo pikeun ngulik métabolisme kolesterol. |
CPDA601447 | PF07328948 | PF-07328948 mangrupa BDK (branched chain keton dehydrogenase kinase) inhibitor oral éféktif. |
CPD112881 | (1S)-2,2,2-trifluoro-1-métilétil]hidrazin hyd... | |
CPD108261 | LOXO-305; LY 3527727; Pirtobrutinib | Pirtobrutinib (LOXO-305) mangrupikeun inhibitor BTK generasi anu selektif pisan sareng non kovalén anu tiasa ngahambat rupa-rupa mutasi substitusi BTK C481. |
CPD115335 | Luxdegalutamide; ARV-766 | Luxdegalutamide (ARV-766) mangrupikeun hidrolisis protéin sasaran chimeric (PROTAC) anu épéktip sacara lisan anu nargétkeun reséptor androgén (AR), anu tiasa nguraikeun mutan résistansi AR. |
CPDA601356 | iHSP110-33 | |
CPDP800487 | TNG462 | TNG-462 mangrupa inhibitor PRMT5 selektif oral éféktif. |
CPDP801649 | 1,2,4-Triazolo[4,3-c]pirimidin-5,8-diamina, N5... | EED ligan 1 mangrupakeun inhibitor rupa-rupa tur éféktif nu nargétkeun subunit EED of methyltransferase PRC2. |
CPDM400208 | 6,7-Difluoro-4 (3H) -quinazolinone | |
CPDP801752 | N-(4-kuinolinilkarbonil)Glisin | |
CPDM400190 | Métil 5-bromo-2-métil-3-(trifluorométil)benz... | |
CPDP800126 | IDE397 (GSK-4362676) | |
CPDP801185 | NST-628 | NST-628 mangrupikeun gél molekular jalur MAPK kalayan perméabilitas panghalang getih-otak, anu tiasa ngahambat fosforilasi RAF sareng aktivasina MEK. |
CPD115153 | NX-2127 | NX-2127 mangrupa inhibitor BTK oral éféktif. |