PI3K

PUSI # Igoa Oloa Fa'amatalaga
CPD1573 GDC-0077 GDC-0077 ose PI3K inhibitor avanoa tautala ma gaioiga antineoplastic ono mafai.
CPD1022 IPI-549 IPI549 o se PI3Kγ Inhibitor malosi ma filifilia ma se IC50 o le 16 nM.
CPDD3857 GDC-0326 GDC-0326 o se inhibitor malosi ma filifili ole α-Isoform o Phosphoinositide 3-Kinase (PI3Kalpha inhibitor). GDC-0326 ausia se maualuga maualuga maualuga o le filifilia i luga o isi kinases. GDC-0326 e maualalo le plasma CL ile tagata.
CPDB0202 AZD8186 AZD8186 o loʻo ma le inhibitor ole beta isoform o le phosphoinositide-3 kinase (PI3K), faʻatasi ai ma gaioiga antineoplastic.
CPDB1536 PQR530 PQR530 o se fa'atosina lua pan-PI3K/mTORC1/2 sili ona malosi.
CPDB1573 GDC-0077 O le GDC-0077 o se fa'aitaga PI3K e avanoa tautala ma filifili (IC50 = 0.038 + 0.003 nM) fa'atasi ai ma> 300-filifili filifilia i luga o isi Vasega I PI3K isoforms.
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