SYK

PUSI # Igoa Oloa Fa'amatalaga
CPDD3529 PRT-060318; PRT318; P142–76 PRT060318 o se inhibitor malosi ma filifili ole spleen tyrosine kinase (Syk; IC50 = 4 nM) .E filifilia, faʻalavelaveina le 92% o le gaioiga Syk, ae o isi kinases o loʻo taofia le> 70% gaioiga, i le faʻatonuga o le 50 nM i se laulau o 270 kinase.
CPDD1851 FAIGA 61-3606 2HCl BAY 61-3606 o se malosi malosi (Ki = 7.5 nM) ma le faʻaiʻuga filifilia o Syk kinase.
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