CAT # | Ingoa Hua | Whakaahuatanga |
CPD111306 | 7-bromo-2,4,6-trichloro-8-fluoroquinazoline | |
CPD113109 | ARS-1323-Alkyne | Ko te ARS-1323-alkyne, he aukati-II pute (S-IIP) aukati |
CPDP801183 | VVD-214;RO7589831;VVD-133214 | Ko te VVD-214 he WRN helicase te aukati allosteric whakamate. |
CPDP801366 | Inlexisertib;DCC-3116 | Ko te DCC-3116 he aukati ULK1/2-waha. |
CPDA601378 | Nonylacridine Orange | |
CPD112537 | 4H-1,3-Dioxolo[4,5-c]pyrrole-4-carboxylic acid,... | |
CPDP801763 | MC3138 | Ko te MC3138 he kaiwhakaoho SIRT5 whiriwhiri. |
CPDP801758 | Chk1-IN-6 | Ko te Chk1-IN-6 he kaha, he whiriwhiri, he kaiao-a-waha, he aukati kaitono CHK1. |
CPD113410 | NDI-101150 | Ko te NDI-101150 he aukati kaha me te whiriwhiri o te HPK1 (hematopoietic progenitor cell kinase 1). |
CPDA601453 | BMS-986408 | Ko te BMS-986408 he aukati DGK α/Zeta rua. |
CPDA601445 | AZD0780;EX-A6975;laroprovstatum; laroprovstat | Ko te PCSK9-IN-12 he pūhui heteroaromatic. Ko te PCSK9-IN-12 he hononga hono mo PCSK9 me te uara Kd<200 nM. Ka taea te whakamahi PCSK9-IN-12 mo te ako o te cholesterol metabolism. |
CPDA601447 | PF07328948 | Ko te PF-07328948 he aukati BDK (ketone dehydrogenase kinase) whai hua-a-waha. |
CPD112881 | (1S)-2,2,2-trifluoro-1-methylethyl]hydrazine hydrazine... | |
CPD108261 | LOXO-305;LY 3527727;Pirtobrutinib | Ko te Pirtobrutinib (LOXO-305) he tino whiriwhiri me te kore covalent muri-whakatupuranga aukati BTK e taea tautāwhi i ngā rerekētanga whakakapinga BTK C481. |
CPD115335 | Luxdegalutamide; ARV-766 | Ko te Luxdegalutamide (ARV-766) he huanga-a-waha e whai hua ana ki te hydrolysis pūmua chimeric (PROTAC) e aro ana ki te kaiwhakawhiwhi androgen (AR), ka taea te whakaheke i nga mutants e pa ana ki te AR. |
CPDA601356 | iHSP110-33 | |
CPDP800487 | TNG462 | Ko te TNG-462 he aukati PRMT5 whai hua ma te waha. |
CPDP801649 | 1,2,4-Triazolo[4,3-c]pyrimidine-5,8-diamine, N5... | Ko te EED ligand 1 he aukati kanorau me te whai hua e aro ana ki te waahanga EED o te methyltransferase PRC2. |
CPDM400208 | 6,7-Difluoro-4(3H)-quinazolinone | |
CPDP801752 | N-(4-quinolinylcarbonyl)Glycine | |
CPDM400190 | Methyl 5-bromo-2-methyl-3-(trifluoromethyl)benz... | |
CPDP800126 | IDE397 (GSK-4362676) | |
CPDP801185 | NST-628 | Ko te NST-628 he MAPK molecular gel me te uruhanga arai toto-roro, ka taea te aukati i te phosphorylation RAF me te whakahohe MEK. |
CPD115153 | NX-2127 | Ko te NX-2127 he aukati BTK whai hua. |