STING

Ologbo # Orukọ ọja Apejuwe
CPD101235 diABZI STING agonist-1 trihydrochloride diABZI STING agonist-1 (trihydrochloride) jẹ apaniyan yiyan ti awọn jiini interferon (STING) agonist olugba, pẹlu EC50s ti 130, 186 nM fun eniyan ati asin, lẹsẹsẹ.
CPD101234 diABZI STING agonist-1 (Tautomerism) diABZI STING agonist-1 Tautomerism (compound 3) jẹ apaniyan yiyan ti awọn jiini interferon (STING) agonist olugba, pẹlu EC50s ti 130, 186 nM fun eniyan ati asin, lẹsẹsẹ.
CPD101233 diABZI STING agonist-1 diABZI STING agonist-1 jẹ oludaniloju yiyan ti awọn jiini interferon (STING) agonist olugba olugba, pẹlu EC50s ti 130, 186 nM fun eniyan ati asin, lẹsẹsẹ.
CPD101232 OGUN STING-4 STING agonist-4 jẹ ohun iwuri ti Interferon Genes (STING) agonist olugba ti o han gbangba inhibitory igbagbogbo (IC50) ti 20 nM. STING agonist-4 jẹ amidobenzimidazole (ABZI) ti o ni ibatan si ami-ara meji lati ṣẹda ABZI (diABZI) ti o ni asopọ pẹlu imudara imudara si STING ati iṣẹ cellular
CPD101231 OGUN STING-3 STING agonist-3, ti a fa jade lati itọsi WO2017175147A1 (apẹẹrẹ 10), jẹ yiyan ati ti kii-nucleotide kekere-moleku STING agonist pẹlu pEC50 ati pIC50 ti 7.5 ati 9.5, lẹsẹsẹ. STING agonist-3 ni ipa egboogi-tumor ti o tọ ati agbara nla lati ni ilọsiwaju itọju ti akàn
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