Awọn ọja

Ologbo # Orukọ ọja Apejuwe
CPD111306 7-bromo-2,4,6-trichloro-8-fluoroquinazoline
CPD113109 ARS-1323-Alkyne ARS-1323-alkyne, a yipada-II apo (S-IIP) onidalẹkun
CPDP801183 VVD-214; RO7589831; VVD-133214 VVD-214 jẹ apaniyan allosteric apaniyan WRN sintetiki.
CPDP801366 Inlexisertib; DCC-3116 DCC-3116 jẹ oludena ULK1/2 ti n ṣiṣẹ ni ẹnu.
CPDA601378 Nonylacridine ọsan
CPD112537 4H-1,3-Dioxolo [4,5-c] pyrrole-4-carboxylic acid,...
CPDP801763 MC3138 MC3138 ni a yan SIRT5 activator.
CPDP801758 Chk1-IN-6 Chk1-IN-6 jẹ oludaniloju oludije CHK1 ti o lagbara, yiyan, ati ẹnu bioavailable.
CPD113410 NDI-101150 NDI-101150 jẹ apaniyan ti o lagbara ati yiyan ti HPK1 (hematopoietic progenitor cell kinase 1).
CPDA601453 BMS-986408 BMS-986408 jẹ imunadoko ẹnu meji DGK α/Zeta inhibitor.
CPDA601445 AZD0780;EX-A6975;laroprovstatum; laroprovstat PCSK9-IN-12 jẹ akojọpọ heteroaromatic kan. PCSK9-IN-12 ni ibaramu abuda fun PCSK9 pẹlu iye Kd kan<200 nM. PCSK9-IN-12 le ṣee lo fun iwadi ti iṣelọpọ idaabobo awọ.
CPDA601447 PF07328948 PF-07328948 jẹ imunadoko ẹnu BDK (ẹka pq ketone dehydrogenase kinase) inhibitor.
CPD112881 (1S) -2,2,2-trifluoro-1-methylethyl]hydrazine hy...
CPD108261 LOXO-305; LY 3527727; Pirtobrutinib Pirtobrutinib (LOXO-305) jẹ yiyan ti o ga pupọ ati inhibitor BTK iran-tẹle ti o le ṣe idiwọ ọpọlọpọ awọn iyipada iyipada BTK C481.
CPD115335 Luxdegalutamide; ARV-766 Luxdegalutamide (ARV-766) jẹ amuaradagba hydrolysis ti o munadoko ti ẹnu si chimeric (PROTAC) ti o fojusi olugba androgen (AR), eyiti o le dinku awọn ẹda ti o ni ibatan AR resistance.
CPDA601356 iHSP110-33
CPDP800487 TNG462 TNG-462 jẹ oludena PRMT5 yiyan ti ẹnu ti o munadoko.
CPDP801649 1,2,4-Triazolo[4,3-c] pyrimidine-5,8-diamine, N5... EED ligand 1 jẹ onidalẹkun oniruuru ati imunadoko ti o dojukọ ipin EED ti methyltransferase PRC2.
CPDM400208 6,7-Difluoro-4 (3H) -quinazolinone
CPDP801752 N- (4-quinolinylcarbonyl) Glycine
CPDM400190 Methyl 5-bromo-2-methyl-3- (trifluoromethyl) benz...
CPDP800126 IDE397 (GSK-4362676)
CPDP801185 NST-628 NST-628 jẹ jeli molikula ipa ọna MAPK pẹlu agbara idena ọpọlọ-ẹjẹ, eyiti o le ṣe idiwọ phosphorylation RAF ati imuṣiṣẹ MEK.
CPD115153 NX-2127 NX-2127 jẹ oludena BTK ti o munadoko ti ẹnu.
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