PI3K

Ologbo # Orukọ ọja Apejuwe
CPD1573 GDC-0077 GDC-0077 jẹ inhibitor PI3K ti o wa ni ẹnu pẹlu iṣẹ ṣiṣe antineoplastic ti o pọju.
CPD1022 IPI-549 IPI549 jẹ oludaniloju PI3Kγ ti o lagbara ati yiyan pẹlu IC50 ti 16 nM.
CPDD3857 GDC-0326 GDC-0326 jẹ oludena ti o lagbara ati yiyan ti α-Isoform of Phosphoinotide 3-Kinase (pi3Kalpha inhibitor). GDC-0326 ṣe aṣeyọri ipele giga pupọ ti yiyan lori awọn kinases miiran. GDC-0326 ni pilasima CL kekere ninu eniyan.
CPDB0202 AZD8186 AZD8186 jẹ ati inhibitor ti isoform beta ti phosphoinotide-3 kinase (PI3K), pẹlu iṣẹ ṣiṣe antineoplastic ti o pọju.
CPDB1536 PQR530 PQR530 jẹ oludena pan-PI3K/mTORC1/2 meji ti o lagbara pupọ.
CPDB1573 GDC-0077 GDC-0077 jẹ ẹnu ti o wa ni ẹnu ati yiyan PI3K inhibitor (IC50 = 0.038 + 0.003 nM) pẹlu> 300-agbo yiyan lori awọn isoforms Kilasi I PI3K miiran.
o

Pe wa

Ìbéèrè

Awọn irohin tuntun

WhatsApp Online iwiregbe!
Close