PI3K

CAT # Product Name Tsanangudzo
CPD1573 GDC-0077 GDC-0077 ndeyemuromo inowanikwa PI3K inhibitor ine inogona kuita antineoplastic chiitiko.
CPD1022 IPI-549 IPI549 ine simba uye inosarudza PI3Kγ Inhibitor ine IC50 ye16 nM.
CPDD3857 GDC-0326 GDC-0326 ine simba uye inosarudza inhibitor ye α-Isoform yePhosphoinositide 3-Kinase (PI3Kalpha inhibitor). GDC-0326 inosvika padanho repamusoro rekusarudza pane mamwe kinase. GDC-0326 ine low plasma CL mumunhu.
CPDB0202 AZD8186 AZD8186 iri uye inhibitor ye beta isoform ye phosphoinositide-3 kinase (PI3K), ine inogona kuita antineoplastic chiitiko.
CPDB1536 PQR530 PQR530 ine simba kwazvo mbiri mbiri pan-PI3K/mTORC1/2 inhibitor.
CPDB1573 GDC-0077 GDC-0077 inowanikwa nemuromo uye inosarudza PI3K inhibitor (IC50 = 0.038 + 0.003 nM) ne> 300-fold selective pane mamwe Class I PI3K isoforms.
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