Vardenafil

Nomen chemicum:

2-(2-ethoxy-5-((4-ethylpiperazin-1-yl) sulfonyl) phenyl) -5-methyl-7-propyl-3,5,6,7-tetrahydro-4H-5l4-imidazo[1; 5-a][1,3,5]triazin-4-one

SMILES Code:

O=C(NC(C1=CC(S(O)(N2CCN(CC)CC2)=O)=CC=C1OCC)=N3)[N]4(C)C3=CN(CCC)C4

InChi Code:

InChI=1S/C23H35N6O4S/c1-5-10-27-16-21-24-22(25-23(30)29(21,4)17-27)19-15-18(8-9-20( 19)33-7-3)34(31,32)28-13-11-26(6-2)12-14-28/h8-9,15-16H,5-7,10-14,17H2; 1-4H3,(H,24,25,30).

InChi Key:

UWRWYSQUBZFWPU-UHFFFAOYSA-N

Keyword:

Vardenafil, Levitra, Staxyn, Vivanza, BAV 38-9456, BAV 38-9456, BAY38-9456, 224785-90-4

Solubilitas:Solutum in DMSO

Repono:0 - 4° C pro brevi termino (dies ad hebdomades), vel -20° C ad terminum longum (menses)

Descriptio:

Vardenafil, etiam quae BAV 38-9456 nota est, inhibitor PDE5 adhibitus est ad praesentes functiones tractandas. Vardenafili indicia et indicia contra-inhibitoria eadem sunt ac cum aliis PDE5 inhibitoribus; propinqua est in munere citrate sildenafil (Viagra) et tadalafil (Cialis). Differentia inter moleculum vardenafili et sildenafili citratum est positio atomi nitrogeni et mutatio globi methyl piperazini sildenafili ad globi ethyl. Tadalafil structura ab utroque sildenafili et vardenafili differt. Vardenafili tempus relative breve efficax comparatur cum sed paulo longiore quam scriptor sildenafili.

Target: PDE5