PI3K

CAT # Izina ryibicuruzwa Ibisobanuro
CPD1573 GDC-0077 GDC-0077 ni munzira iboneka ya PI3K inhibitor hamwe nibikorwa bya antineoplastique.
CPD1022 IPI-549 IPI549 ni Inhibitor ikomeye kandi ihitamo PI3Kγ ifite IC50 ya 16 nM.
CPDD3857 GDC-0326 GDC-0326 ni inhibitor ikomeye kandi ihitamo α-Isoform ya Phosphoinositide 3-Kinase (PI3Kalpha inhibitor). GDC-0326 igera kurwego rwo hejuru cyane rwo guhitamo kurenza izindi kinase. GDC-0326 ifite plasma nkeya CL mubantu.
CPDB0202 AZD8186 AZD8186 ni na inhibitor ya beta isoform ya fosifinositide-3 kinase (PI3K), hamwe nibikorwa bya antineoplastique.
CPDB1536 PQR530 PQR530 ninzitizi ikomeye cyane pan-PI3K / mTORC1 / 2 inhibitor.
CPDB1573 GDC-0077 GDC-0077 ni munwa iboneka kandi ihitamo PI3K inhibitor (IC50 = 0.038 + 0.003 nM) hamwe> guhitamo inshuro 300 kurenza ayandi masomo ya I PI3K.
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