SYK

CAT # Izina ryibicuruzwa Ibisobanuro
CPDD3529 PRT-060318; PRT318; P142–76 PRT060318 ninzitizi ikomeye kandi ihitamo inhibitori ya spleen tyrosine kinase (Syk; IC50 = 4 nM) .Birahitamo, bibuza 92% byibikorwa bya Syk, mugihe izindi kinase zigumana> 70%, murwego rwa 50 nM mukibaho 270 kinase.
CPDD1851 BAY 61-3606 2HCl BAY 61-3606 nimbaraga (Ki = 7.5 nM) hamwe na inhibitor ya Syk kinase.
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