Ibicuruzwa

CAT # Izina ryibicuruzwa Ibisobanuro
CPD111306 7-bromo-2,4,6-trichloro-8-fluoroquinazoline
CPD113109 ARS-1323-Alkyne ARS-1323-alkyne, umufuka-II umufuka (S-IIP) inhibitor
CPDP801183 VVD-214; RO7589831; VVD-133214 VVD-214 ni synthique WRN helicase yica allosteric inhibitor.
CPDP801366 Inlexisertib; DCC-3116 DCC-3116 ni umunwa ukora ULK1 / 2 inhibitor.
CPDA601378 Nonylacridine Orange
CPD112537 4H-1,3-Dioxolo [4,5-c] pyrrole-4-acide karubike, ...
CPDP801763 MC3138 MC3138 nuwatoranije SIRT5.
CPDP801758 Chk1-IN-6 Chk1-IN-6 ni imbaraga, guhitamo, no munwa bioavailable CHK1 umukandida inhibitor.
CPD113410 NDI-101150 NDI-101150 ni inzitizi ikomeye kandi ihitamo HPK1 (hematopoietic progenitor selile kinase 1).
CPDA601453 BMS-986408 BMS-986408 ni umunwa mwiza DGK α / Zeta inhibitor.
CPDA601445 AZD0780; EX-A6975; laroprovstatum; laroprovstat PCSK9-IN-12 ni ibice bitandukanye. PCSK9-IN-12 ifite isano ihuza PCSK9 ifite agaciro ka Kd<200 nM. PCSK9-IN-12 irashobora gukoreshwa mukwiga metabolism ya cholesterol.
CPDA601447 PF07328948 PF-07328948 ni umunwa wa BDK (urunigi rwashami ketone dehydrogenase kinase) inhibitor.
CPD112881 (1S) -2,2,2-trifluoro-1-methylethyl] hydrazine hy ...
CPD108261 LOXO-305; LY 3527727; Pirtobrutinib Pirtobrutinib (LOXO-305) ni ihitamo ryinshi kandi ridahwitse ibisekuruza bizaza BTK inhibitor ishobora kubuza ihinduka ryimiterere rya BTK C481.
CPD115335 Luxdegalutamide; ARV-766 Luxdegalutamide (ARV-766) ni poroteyine hydrolysis ikora neza mu kanwa igamije chimeric (PROTAC) yibasira reseptor ya androgene (AR), ishobora gutesha agaciro ihinduka ry’imiterere ya AR.
CPDA601356 iHSP110-33
CPDP800487 TNG462 TNG-462 nuburyo bwiza bwo guhitamo PRMT5 inhibitor.
CPDP801649 1,2,4-Triazolo [4,3-c] pyrimidine-5,8-diamine, N5 ... EED ligand 1 ni inhibitor itandukanye kandi ikora neza yibasira EED subunit ya methyltransferase PRC2.
CPDM400208 6,7-Difluoro-4 (3H) -quinazolinone
CPDP801752 N- (4-quinolinylcarbonyl) Glycine
CPDM400190 Methyl 5-bromo-2-methyl-3- (trifluoromethyl) benz ...
CPDP800126 IDE397 (GSK-4362676)
CPDP801185 NST-628 NST-628 ni inzira ya MAPK inzira ya molekile gel ifite ubwonko bwamaraso n'ubwonko bwinjira, bushobora kubuza RAF fosifora na MEK gukora.
CPD115153 NX-2127 NX-2127 ni imvugo ya BTK ikora neza.
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