SYK

MPAKA # Dzina lazogulitsa Kufotokozera
Chithunzi cha CPDD3529 PRT-060318; PRT318; P142-76 PRT060318 ndi inhibitor yamphamvu komanso yosankha ya spleen tyrosine kinase (Syk; IC50 = 4 nM). Imasankha, imalepheretsa 92% ya zochita za Syk, pamene kinase ena amasunga> 70% ntchito, pamagulu a 50 nM mu gulu la 270 magalamu.
Chithunzi cha CPDD1851 Chithunzi cha BAY 61-3606 2HCl BAY 61-3606 ndi yamphamvu (Ki = 7.5 nM) ndi inhibitor yosankha ya Syk kinase.
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