KUCING # | Jeneng produk | Katrangan |
CPD111306 | 7-bromo-2,4,6-trikloro-8-fluoroquinazoline | |
CPD113109 | ARS-1323-Alkyne | ARS-1323-alkyne, inhibitor switch-II pocket (S-IIP). |
CPDP801183 | VVD-214;RO7589831;VVD-133214 | VVD-214 minangka inhibitor alosterik helikase WRN sintetik. |
CPDP801366 | Inlexisertib;DCC-3116 | DCC-3116 minangka inhibitor ULK1/2 oral aktif. |
CPDA601378 | Oranye Nonylacridine | |
CPD112537 | 4H-1,3-Dioxolo[4,5-c]pirol-4-asam karboksilat,... | |
CPDP801763 | MC3138 | MC3138 minangka aktivator SIRT5 sing selektif. |
CPDP801758 | Chk1-IN-6 | Chk1-IN-6 minangka inhibitor calon CHK1 sing kuat, selektif, lan kasedhiya kanthi lisan. |
CPD113410 | NDI-101150 | NDI-101150 minangka inhibitor HPK1 sing kuat lan selektif (hematopoietic progenitor cell kinase 1). |
CPDA601453 | BMS-986408 | BMS-986408 minangka inhibitor DGK α/Zeta ganda sing efektif sacara lisan. |
CPDA601445 | AZD0780;EX-A6975;laroprovstatum; laroprovstat | PCSK9-IN-12 minangka senyawa heteroaromatik. PCSK9-IN-12 wis naleni karemenan kanggo PCSK9 karo nilai Kd<200 nM. PCSK9-IN-12 bisa digunakake kanggo sinau metabolisme kolesterol. |
CPDA601447 | PF07328948 | PF-07328948 minangka inhibitor BDK (branched chain ketone dehydrogenase kinase) sing efektif sacara lisan. |
CPD112881 | (1S)-2,2,2-trifluoro-1-methylethyl]hydrazine h... | |
CPD108261 | LOXO-305;LY 3527727;Pirtobrutinib | Pirtobrutinib (LOXO-305) minangka inhibitor BTK generasi sabanjure sing paling selektif lan non kovalen sing bisa nyandhet macem-macem mutasi substitusi BTK C481. |
CPD115335 | Luxdegalutamide; ARV-766 | Luxdegalutamide (ARV-766) minangka chimeric target hidrolisis protein sing efektif sacara lisan (PROTAC) sing nargetake reseptor androgen (AR), sing bisa ngrusak mutan sing gegandhengan karo resistensi AR. |
CPDA601356 | iHSP110-33 | |
CPDP800487 | TNG462 | TNG-462 minangka inhibitor PRMT5 selektif sing efektif sacara lisan. |
CPDP801649 | 1,2,4-Triazolo[4,3-c]pirimidin-5,8-diamine, N5... | EED ligan 1 minangka inhibitor macem-macem lan efektif sing target subunit EED saka methyltransferase PRC2. |
CPDM400208 | 6,7-Difluoro-4 (3H) -quinazolinone | |
CPDP801752 | N-(4-quinolinylcarbonyl)Glycine | |
CPDM400190 | Metil 5-bromo-2-metil-3-(trifluoromethyl)benz... | |
CPDP800126 | IDE397 (GSK-4362676) | |
CPDP801185 | NST-628 | NST-628 minangka gel molekul jalur MAPK kanthi permeabilitas penghalang getih-otak, sing bisa nyandhet fosforilasi RAF lan aktivasi MEK. |
CPD115153 | NX-2127 | NX-2127 minangka inhibitor BTK sing efektif sacara lisan. |