KAT # | Produkt Namme | Beskriuwing |
CPD111306 | 7-bromo-2,4,6-trichloro-8-fluoroquinazoline | |
CPD113109 | ARS-1323-Alkyne | ARS-1323-alkyn, in switch-II pocket (S-IIP) inhibitor |
CPDP801183 | VVD-214;RO7589831;VVD-133214 | VVD-214 is in syntetyske WRN helicase deadlike allosteryske inhibitor. |
CPDP801366 | Inlexisertib;DCC-3116 | DCC-3116 is in oraal aktive ULK1/2-ynhibitor. |
CPDA601378 | Nonylacridine Oranje | |
CPD112537 | 4H-1,3-Dioxolo[4,5-c]pyrrol-4-carboxylic acid, ... | |
CPDP801763 | MC3138 | MC3138 is in selektyf SIRT5 activator. |
CPDP801758 | Chk1-IN-6 | Chk1-IN-6 is in krêftige, selektive en oraal biobeskikbere CHK1 kandidaat-inhibitor. |
CPD113410 | NDI-101150 | NDI-101150 is in krêftige en selektive ynhibitor fan HPK1 (hematopoietic progenitor cell kinase 1). |
CPDA601453 | BMS-986408 | BMS-986408 is in oraal effektive dûbele DGK α / Zeta inhibitor. |
CPDA601445 | AZD0780;EX-A6975;laroprovstatum; laroprovstat | PCSK9-IN-12 is in heteroaromatyske ferbining. PCSK9-IN-12 hat binende affiniteit foar PCSK9 mei in Kd wearde<200 nM. PCSK9-IN-12 kin brûkt wurde foar de stúdzje fan cholesterolmetabolisme. |
CPDA601447 | PF07328948 | PF-07328948 is in oraal effektive BDK (branched chain ketone dehydrogenase kinase) inhibitor. |
CPD112881 | (1S)-2,2,2-trifluor-1-methylethyl]hydrazine hy... | |
CPD108261 | LOXO-305;LY 3527727;Pirtobrutinib | Pirtobrutinib (LOXO-305) is in heul selektive en net-kovalente BTK-ynhibitor fan folgjende generaasje dy't ferskate BTK C481-substitúsjonele mutaasjes kin remme. |
CPD115335 | Luxdegalutamide; ARV-766 | Luxdegalutamide (ARV-766) is in oraal effektive proteïnehydrolyse-targete chimeric (PROTAC) targeting androgen receptor (AR), dy't AR-resistinsje relatearre mutanten kin degradearje. |
CPDA601356 | iHSP110-33 | |
CPDP800487 | TNG462 | TNG-462 is in mûnling effektive selektive PRMT5-ynhibitor. |
CPDP801649 | 1,2,4-triazolo[4,3-c]pyrimidine-5,8-diamine, N5... | EED ligand 1 is in ferskaat en effektive ynhibitor dy't rjochtet op de EED subunit fan methyltransferase PRC2. |
CPDM400208 | 6,7-Difluoro-4(3H)-kinazolinone | |
CPDP801752 | N-(4-kinolinylkarbonyl)glycine | |
CPDM400190 | Methyl 5-bromo-2-methyl-3-(trifluormethyl)benz... | |
CPDP800126 | IDE397 (GSK-4362676) | |
CPDP801185 | NST-628 | NST-628 is in MAPK-paad molekulêre gel mei permeabiliteit fan bloed-harsensbarriêre, dy't RAF-fosforylaasje en MEK-aktivearring kin remme. |
CPD115153 | NX-2127 | NX-2127 is in oraal effektive BTK-ynhibitor. |