PI3K

CAT # Igama lemveliso Inkcazo
CPD1573 GDC-0077 I-GDC-0077 yi-PI3K inhibitor ekhoyo ngomlomo enokuthi ibe nomsebenzi we-antineoplastic.
CPD1022 IPI-549 I-IPI549 inamandla kwaye ikhetha i-PI3Kγ Inhibitor ene-IC50 ye-16 nM.
CPDD3857 GDC-0326 I-GDC-0326 yi-inhibitor enamandla kwaye ekhethiweyo ye-α-Isoform ye-Phosphoinositide 3-Kinase (PI3Kalpha inhibitor). I-GDC-0326 ifikelela kwinqanaba eliphezulu kakhulu lokukhetha ngaphezu kwezinye i-kinases. I-GDC-0326 ine-plasma ephantsi ye-CL emntwini.
CPDB0202 I-AZD8186 I-AZD8186 kunye ne-inhibitor ye-beta isoform ye-phosphoinositide-3 kinase (PI3K), kunye nomsebenzi onokuthi ube ne-antineoplastic.
CPDB1536 PQR530 I-PQR530 yi-dual inhibitor enamandla kakhulu-PI3K/mTORC1/2.
CPDB1573 GDC-0077 I-GDC-0077 ifumaneka ngomlomo kwaye ikhethiweyo ye-PI3K inhibitor (IC50 = 0.038 + 0.003 nM) kunye> 300-fold selective over other Class I PI3K isoforms.

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