EGFR

KATSE # Lebitso la Sehlahiswa Tlhaloso
CPD100230 JBJ-04-125-02 R-isomer
CPD3232 NTN21277 NTN21277, e tsejoang hape ka hore ke PROTAC 3 e thehiloeng ho Gefitinib ke VHL-recruiting PROTAC e bakang ho senyeha ha liphetoho tsa EGFR le EGFR ka DC50 ea 11.7 nM le 22.3 nM bakeng sa lisele tsa HCC827 (Exon 19 del) le H3255 cell (L8258).
CPDB3615 Nazartinib; EGF816; NVS-816 Nazartinib, eo hape e tsejoang e le EGF816 le NVS-816, ke inhibitor e fumanehang ka molomo, e ke keng ea fetoloa, ea moloko oa boraro, e khethiloeng ke epidermal growth factor receptor (EGFR) inhibitor, e nang le ts'ebetso e ka bang teng ea antineoplastic.
CPDB0934 EAI-045 EAI045 e matla le e khethang ea EGFR inhbitor. EAI045 e ikemiselitse ho khetha liphetoho tsa EGFR tse hananang le lithethefatsi empa e boloka moamoheli oa mofuta o hlaha. EAI045 e thibela EGFR ea L858R/T790M-mutant e nang le matla a tlase a nanomolar litekong tsa biochemical.
CPDB0101 Poziotinib Mefuta e nang le poziotinib e ntse e etsoa lipatlisiso litekong tsa meriana bakeng sa phekolo ea EGFR-mutant lung adenocarcinoma.
CPDB0137 Osimertinib Mesylate Osimertinib, eo hape e tsejoang e le mereletinib le AZD-9291, ke moloko oa boraro oa EGFR inhibitor, o bontšitse tšepiso lithutong tsa pele ho nako 'me o fana ka tšepo ho bakuli ba nang le kankere ea matšoafo e tsoetseng pele e seng e hanyetsana le li-inhibitors tsa EGFR tse teng.
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