TANGI

CAT # Ingoa Hua Whakaahuatanga
CPD101235 diABZI STING agonist-1 trihydrochloride Ko te diABZI STING agonist-1 (trihydrochloride) he kaiwhakatairanga whiriwhiri o nga ira interferon (STING) kaiwhakawhiwhi agonist, me nga EC50 o 130, 186 nM mo te tangata me te kiore, ia.
CPD101234 diABZI STING agonist-1 (Tautomerism) diABZI STING agonist-1 Tautomerism (compound 3) is a selective stimulator of interferon genes (STING) receptor agonist, with EC50s of 130, 186 nM mo te tangata me te kiore, ia.
CPD101233 diABZI STING agonist-1 Ko te diABZI STING agonist-1 he kaiwhakatairanga maataki o nga ira interferon (STING) kaiawhina agonist, me nga EC50 o 130, 186 nM mo te tangata me te kiore.
CPD101232 STING agonist-4 Ko te STING agonist-4 he kaiwhakatairanga o te Interferon Genes (STING) agonist kaiawhina me te kaha aukati (IC50) o te 20 nM. Ko te STING agonist-4 he pūhui hangarite e rua-a-amidobenzimidazole (ABZI) hei hanga i nga ABZI hono (diABZI) me te pai ake o te here ki te STING me te mahi pūkoro.
CPD101231 STING agonist-3 Ko te STING agonist-3, he mea tango mai i te patent WO2017175147A1 (tauira 10), he agonist STING iti-mucleotide iti me te pEC50 me te pIC50 o te 7.5 me te 9.5, ia. Ko te STING agonist-3 he awenga aukati-puku mauroa me te kaha nui ki te whakapai ake i te maimoatanga o te mate pukupuku
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