STING

KUCING # Jeneng produk Katrangan
CPD101235 diABZI STING agonis-1 trihidroklorida diABZI STING agonist-1 (trihydrochloride) minangka stimulator selektif saka gen interferon (STING) reseptor agonis, kanthi EC50s 130, 186 nM kanggo manungsa lan tikus, masing-masing.
CPD101234 diABZI STING agonist-1 (Tautomerism) diABZI STING agonist-1 Tautomerism (senyawa 3) minangka stimulator selektif saka gen interferon (STING) reseptor agonis, kanthi EC50s saka 130, 186 nM kanggo manungsa lan mouse, mungguh.
CPD101233 diaABZI STING agonis-1 diABZI STING agonist-1 minangka stimulator selektif saka agonis reseptor gen interferon (STING), kanthi EC50s 130, 186 nM kanggo manungsa lan tikus.
CPD101232 STING agonis-4 Agonis STING-4 minangka stimulator saka agonis reseptor Interferon Genes (STING) kanthi konstanta inhibisi sing jelas (IC50) 20 nM. STING agonis-4 minangka senyawa adhedhasar amidobenzimidazole (ABZI) sing gegandhengan karo simetri kanggo nggawe ABZIs (diABZIs) sing disambungake kanthi ikatan sing luwih apik kanggo STING lan fungsi seluler.
CPD101231 STING agonis-3 STING agonist-3, diekstrak saka paten WO2017175147A1 (conto 10), minangka agonis STING molekul cilik sing selektif lan non-nukleotida kanthi pEC50 lan pIC50 saka 7,5 lan 9,5. STING agonist-3 nduweni efek anti-tumor sing tahan lama lan potensial banget kanggo ningkatake perawatan kanker
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