SYK

nwamba # Aha ngwaahịa Nkọwa
CPDD3529 PRT-060318; PRT318; P142–76 PRT060318 bụ onye na-eme ihe ike ma na-ahọrọ nke spleen tyrosine kinase (Syk; IC50 = 4 nM) .Ọ bụ nhọrọ, na-egbochi 92% nke ọrụ Syk, ebe ndị ọzọ kinases na-ejigide>70% ọrụ, na ntinye nke 50 nM na panel panel nke. 270 ụdị.
CPDD1851 BAY 61-3606 2HCl BAY 61-3606 bụ onye nwere ike (Ki = 7.5 nM) yana onye na-egbochi Syk kinase.
nke

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