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CHAT # Non pwodwi Deskripsyon
CPD111306 7-bromo-2,4,6-trichloro-8-fluoroquinazoline
CPD113109 ARS-1323-Alkyne ARS-1323-alkyne, yon pòch switch-II (S-IIP) inhibiteur
CPDP801183 VVD-214;RO7589831;VVD-133214 VVD-214 se yon inibitè alosterik letal WRN helicase sentetik.
CPDP801366 Inlexisertib;DCC-3116 DCC-3116 se yon inibitè ULK1/2 aktif oralman.
CPDA601378 Nonylacridine zoranj
CPD112537 4H-1,3-Dioxolo[4,5-c]pyrrole-4-carboxylic asid,...
CPDP801763 MC3138 MC3138 se yon activator selektif SIRT5.
CPDP801758 Chk1-IN-6 Chk1-IN-6 se yon inibitè kandida CHK1 ki pisan, selektif ak oral byodisponib.
CPD113410 NDI-101150 NDI-101150 se yon inibitè ki pisan ak selektif nan HPK1 (ematopoietic progenitor selil kinaz 1).
CPDA601453 BMS-986408 BMS-986408 se yon oralman efikas doub DGK α/Zeta inibitè.
CPDA601445 AZD0780;EX-A6975;laroprovstatum; laroprovstat PCSK9-IN-12 se yon konpoze heteroaromatic. PCSK9-IN-12 gen afinite obligatwa pou PCSK9 ak yon valè Kd<200 nM. PCSK9-IN-12 ka itilize pou etid metabolis kolestewòl.
CPDA601447 PF07328948 PF-07328948 se yon inibitè oralman efikas BDK (branche chèn keton dehydrogenase kinase).
CPD112881 (1S) -2,2,2-trifluoro-1-methylethyl]hydrazine hy...
CPD108261 LOXO-305;LY 3527727;Pirtobrutinib Pirtobrutinib (LOXO-305) se yon inibitè BTK trè selektif ak ki pa kovalan nan pwochen jenerasyon ki ka anpeche divès kalite mitasyon sibstitisyon BTK C481.
CPD115335 Luxdegalutamid; ARV-766 Luxdegalutamide (ARV-766) se yon oralman efikas idroliz pwoteyin vize chimerik (PROTAC) vize reseptè androjèn (AR), ki ka degrade mutan ki gen rapò ak rezistans AR.
CPDA601356 iHSP110-33
CPDP800487 TNG462 TNG-462 se yon inibitè PRMT5 selektif oralman efikas.
CPDP801649 1,2,4-Triazolo [4,3-c] pirimidin-5,8-diamine, N5... EED ligand 1 se yon inibitè divès ak efikas ki vize sou-inite EED nan methyltransferase PRC2.
CPDM400208 6,7-Difluoro-4 (3H)-quinazolinone
CPDP801752 N-(4-quinolinylcarbonyl)Glycine
CPDM400190 Methyl 5-bromo-2-methyl-3-(trifluorometil)benz...
CPDP800126 IDE397 (GSK-4362676)
CPDP801185 NST-628 NST-628 se yon jèl molekilè MAPK ak pèmeyabilite baryè san-sèvo, ki ka anpeche fosforilasyon RAF ak aktivasyon MEK.
CPD115153 NX-2127 NX-2127 se yon inibitè BTK oralman efikas.

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