SYK

CAT # Sunan samfur Bayani
Saukewa: CPDD3529 PRT-060318; PRT318; P142-76 PRT060318 shine mai hanawa mai ƙarfi da zaɓi na spleen tyrosine kinase (Syk; IC50 = 4 nM) . Yana da zaɓi, yana hana 92% na aikin Syk, yayin da sauran kinases suna riƙe> 70% aiki, a wani taro na 50 nM a cikin wani panel na 270 kinsa.
Saukewa: CPDD1851 BAY 61-3606 2HCl BAY 61-3606 mai ƙarfi ne (Ki = 7.5 nM) kuma mai hanawa na Syk kinase.
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