MI

KATSE # Lebitso la Sehlahiswa Tlhaloso
CPD3218 BMS-955176 GSK3532795, e tsejoang hape e le BMS-955176, ke sehlahisoa se matla, se sebetsang ka molomo, sa moloko oa bobeli sa HIV-1 maturation inhibitor (MI) se tsoetseng pele ka liteko tsa kliniki tsa phase IIb. GSK3532795 e kopanya tšireletso e pharaletseng ea likokoana-hloko tsa polymorphic (EC50<15 nM ho sehlopha sa lipolymorphisms tse tloaelehileng tse emelang 96.5% HIV-1 subtype B virus) e nang le profil e ntle ea pharmacokinetic mefuteng ea preclinical.
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