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KATSE # Lebitso la Sehlahiswa Tlhaloso
CPD101235 diABZI STING agonist-1 trihydrochloride diABZI STING agonist-1 (trihydrochloride) ke stimulator e khethollang ea liphatsa tsa lefutso tsa interferon (STING) receptor agonist, e nang le EC50s ea 130, 186 nM bakeng sa motho le mouse, ka ho latellana.
CPD101234 diABZI STING agonist-1 (Tautomerism) diABZI STING agonist-1 Tautomerism (motsoako oa 3) ke ntho e susumetsang e khethollang ea liphatsa tsa lefutso tsa interferon (STING) receptor agonist, e nang le EC50s ea 130, 186 nM bakeng sa motho le mouse, ka ho latellana.
CPD101233 diABZI STING agonist-1 diABZI STING agonist-1 ke ntho e susumetsang e khethollang ea liphatsa tsa lefutso tsa interferon (STING), tse nang le EC50s ea 130, 186 nM bakeng sa motho le mouse, ka ho latellana.
CPD101232 STING agonist-4 STING agonist-4 ke stimulator ea Interferon Genes (STING) receptor agonist e nang le inhibitory constant (IC50) ea 20 nM. STING agonist-4 ke metsoako e 'meli e amanang le amidobenzimidazole (ABZI) e amanang le symmetry ho theha li-ABZI tse hokahantsoeng (diABZIs) tse nang le tlamo e matlafalitsoeng ho STING le tšebetso ea cellular.
CPD101231 STING agonist-3 STING agonist-3, e ntšitsoeng ho patent WO2017175147A1 (mohlala 10), ke ntho e khethollang le e seng ea nucleotide e nyenyane ea molek'hule STING agonist e nang le pEC50 le pIC50 ea 7.5 le 9.5, ka ho latellana. STING agonist-3 e na le phello e tšoarellang ea anti-tumor le monyetla o moholo oa ho ntlafatsa kalafo ea mofets'e
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