86-21-64556180 ib

MI

CAT # Khoom npe Kev piav qhia
PEB 3218 BMS-955176 GSK3532795, tseem hu ua BMS-955176, yog lub zog, qhov ncauj nquag, thib ob tiam HIV-1 maturation inhibitor (MI) uas tau nce mus txog theem IIb kev sim tshuaj. GSK3532795 sib txuas dav dav ntawm cov kab mob polymorphic (EC50)<15 nM mus rau lub vaj huam sib luag ntawm cov neeg sawv cev ntawm ntau hom polymorphisms ntawm 96.5% HIV-1 subtype B tus kab mob) nrog rau cov tshuaj pharmacokinetic profile nyob rau hauv hom preclinical.
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